摘要 |
<P>PROBLEM TO BE SOLVED: To provide diaryl-purines, -azapurines and -deazapurines as non-nucleoside reverse transcriptase inhibitors. <P>SOLUTION: The invention concerns 2-phenylamino-6-aryl amino-, 6-aryloxy-, and 6- arylthio- purines, -azapurines and -deazapurines. The compounds are non-nucleoside reverse transcriptase inhibitors and have potential as anti-HIV treatment. <P>COPYRIGHT: (C)2013,JPO&INPIT |