发明名称 DIARYL-PURINE, -AZAPURINE AND -DEAZAPURINE AS NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS FOR TREATMENT OF HIV
摘要 <P>PROBLEM TO BE SOLVED: To provide diaryl-purines, -azapurines and -deazapurines as non-nucleoside reverse transcriptase inhibitors. <P>SOLUTION: The invention concerns 2-phenylamino-6-aryl amino-, 6-aryloxy-, and 6- arylthio- purines, -azapurines and -deazapurines. The compounds are non-nucleoside reverse transcriptase inhibitors and have potential as anti-HIV treatment. <P>COPYRIGHT: (C)2013,JPO&INPIT
申请公布号 JP2012188454(A) 申请公布日期 2012.10.04
申请号 JP20120143245 申请日期 2012.06.26
申请人 ARDEA BIOSCIENCES INC 发明人 GIRARDET JEAN LUC;KOH YUNG-HYO;SHAW STEPHANIE;KIM HONG WOO
分类号 A61K31/519;A61P31/18;C07D487/04 主分类号 A61K31/519
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