发明名称 |
METHOD FOR PRODUCING BENZYLPYRAZOLE DERIVATIVE AND PRODUCTION INTERMEDIATE THEREOF |
摘要 |
A production intermediate of a glucopyranosyloxypyrazole derivative which is represented by general formula (E) (wherein R3 and R4 are as defined below) and is useful as a therapeutic agent for diabetes or the like, and a method for producing a benzylpyrazole derivative, said method being indistrially more advantageous than conventional methods for producing a benzylpyrazole derivative, can be provided by causing a reaction of a compound represented by general formula (D) (wherein each of R1 and R2 represents a C1-6 alkyl group or the like; R3 represents a halogen atom, a C1-6 alkoxy group or the like; and R4 represents a hydrogen atom, a halogen atom, a C1-6 alkoxy group or the like). |
申请公布号 |
WO2012133783(A1) |
申请公布日期 |
2012.10.04 |
申请号 |
WO2012JP58604 |
申请日期 |
2012.03.30 |
申请人 |
KISSEI PHARMACEUTICAL CO., LTD.;AINAI, TAKAYUKI;KOBAYASHI, MASAHIRO |
发明人 |
AINAI, TAKAYUKI;KOBAYASHI, MASAHIRO |
分类号 |
C07D317/30;C07D231/20 |
主分类号 |
C07D317/30 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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