发明名称 |
DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-a]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES |
摘要 |
Derivatives of 6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid amide exhibit good inhibitory effect upon the interaction of CAMs and Leukointegrins and are thus useful in the treatment of inflammatory disease. |
申请公布号 |
US2012252817(A1) |
申请公布日期 |
2012.10.04 |
申请号 |
US201013375767 |
申请日期 |
2010.05.26 |
申请人 |
LEMIEUX RENE MARC;BRUNETTE STEVEN RICHARD;HORAN JOSHUA COURTNEY;KOWALSKI JENNIFER A.;LAWLOR MICHAEL DAVID;MCKIBBEN BRYAN;MILLER CRAIG ANDREW;BARBOSA ANTONIO J. M.;BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
LEMIEUX RENE MARC;BRUNETTE STEVEN RICHARD;HORAN JOSHUA COURTNEY;KOWALSKI JENNIFER A.;LAWLOR MICHAEL DAVID;MCKIBBEN BRYAN;MILLER CRAIG ANDREW;BARBOSA ANTONIO J. M. |
分类号 |
C07D487/04;A61K31/4439;A61K31/501;A61K31/506;A61P1/00;A61P1/04;A61P3/10;A61P5/16;A61P7/00;A61P9/10;A61P11/00;A61P11/06;A61P13/12;A61P17/00;A61P17/06;A61P19/02;A61P19/04;A61P25/00;A61P27/02;A61P29/00;A61P31/00;A61P37/00;A61P37/06 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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