发明名称 |
ARYL SULPHONE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS |
摘要 |
Methods and compounds effective in ameliorating conditions characterized by unwanted calcium channel activity, particularly unwanted N-type and/or T-type calcium channel activity, are disclosed. Specifically, a series of compounds containing aryl sulphone derivatives, as exemplified by Formula (I).
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申请公布号 |
US2012245137(A1) |
申请公布日期 |
2012.09.27 |
申请号 |
US201013496729 |
申请日期 |
2010.09.17 |
申请人 |
PAJOUHESH HASSAN A.;GALEMMO, JR. ROBERT;HOLLAND RICHARD;ZHOU YUANXI;ZHU YONGBAO;SIMONSON ERIC;CHAHAL NAVJOT;GRIMWOOD MIKE;ZALICUS PHARMACEUTICALS LTD. |
发明人 |
PAJOUHESH HASSAN A.;GALEMMO, JR. ROBERT;HOLLAND RICHARD;ZHOU YUANXI;ZHU YONGBAO;SIMONSON ERIC;CHAHAL NAVJOT;GRIMWOOD MIKE |
分类号 |
A61K31/44;A61K31/166;A61K31/397;A61K31/505;A61K31/5375;A61K31/538;A61P25/00;A61P25/06;A61P25/08;A61P25/16;A61P25/18;A61P25/24;C07C317/48;C07D205/04;C07D213/82;C07D239/26;C07D265/36;C07D295/13 |
主分类号 |
A61K31/44 |
代理机构 |
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