发明名称 FUSED TRICYCLIC DUAL INHIBITORS OF CDK 4/6 AND FLT3
摘要 Compounds of Formula (I) are useful inhibitors of CDK 4, CDK6, and FLT3. Such compounds are useful in treating cancer and various other disease conditions. Compounds of Formula (I) have the following structure: where R1 is a group of Formula (IA), Formula (IB), Formula (IC), or Formula (ID) and the definitions of the other variables are provided herein.
申请公布号 WO2012129344(A1) 申请公布日期 2012.09.27
申请号 WO2012US30007 申请日期 2012.03.21
申请人 AMGEN INC.;CHEN, XIAOQI;DAI, KANG;DUQUETTE, JASON;GRIBBLE, MICHAEL W., JR.;HUARD, JUSTIN N.;KEEGAN, KATHLEEN S.;LI, ZHIHONG;LIVELY, SARAH E.;MCGEE, LAWRENCE R.;RAGAINS, MARK L.;WANG, XIANGHONG;WEIDNER, MARGARET F.;ZHANG, JIAN 发明人 CHEN, XIAOQI;DAI, KANG;DUQUETTE, JASON;GRIBBLE, MICHAEL W., JR.;HUARD, JUSTIN N.;KEEGAN, KATHLEEN S.;LI, ZHIHONG;LIVELY, SARAH E.;MCGEE, LAWRENCE R.;RAGAINS, MARK L.;WANG, XIANGHONG;WEIDNER, MARGARET F.;ZHANG, JIAN
分类号 C07D471/14;A61K31/519;A61P35/00;A61P35/02;C07D519/00 主分类号 C07D471/14
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