发明名称 |
4-methylpyridopyrimidinone compounds |
摘要 |
The present invention is directed to novel 4-methylpyridopyrimidinone compounds of Formula (I), and to salts thereof, their synthesis, and their use as inhibitors of phosphoinositide 3-kinase alpha (PI3-Kα). |
申请公布号 |
US8273755(B2) |
申请公布日期 |
2012.09.25 |
申请号 |
US20100702937 |
申请日期 |
2010.02.09 |
申请人 |
CHENG HENGMIAO;BHUMRALKAR DILIP;DRESS KLAUS RUPRECHT;HOFFMAN JACQUI ELIZABETH;JOHNSON MARY CATHERINE;KANIA ROBERT STEVEN;LE PHUONG THI QUY;NAMBU MITCHELL DAVID;PAIRISH MASON ALAN;PLEWE MICHAEL BRUNO;TRAN KHANH TUAN;PFIZER INC |
发明人 |
CHENG HENGMIAO;BHUMRALKAR DILIP;DRESS KLAUS RUPRECHT;HOFFMAN JACQUI ELIZABETH;JOHNSON MARY CATHERINE;KANIA ROBERT STEVEN;LE PHUONG THI QUY;NAMBU MITCHELL DAVID;PAIRISH MASON ALAN;PLEWE MICHAEL BRUNO;TRAN KHANH TUAN |
分类号 |
C07D471/04;A61K31/519;A61P35/00 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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