发明名称 SALT FORM OF HYDROXYPHENYLALANINE KINASE INHIBITOR
摘要 <p>The present invention pertains to acidic adduct salts of (Z)-N-[2-(diethylamino)ethyl]-2-methyl-7-(1,2-dihydro-5-fluoro-2-oxo-3H-indol-3-ylene)-4,5,6,7-tetrahydro-1H-indol-3-carboxamide, selected from L-malate, hydrochloride, phosphate, L-tartrate, benzene sulfonate, sulfate, methanesulfonate, succinate, citrate, fumarate, p-toluenesulfonate, hydrobromate, L-mandelate, lactate, acetate and maleate, and the use of the above salt compounds for preparing pharmaceuticals.</p>
申请公布号 WO2012122921(A1) 申请公布日期 2012.09.20
申请号 WO2012CN72174 申请日期 2012.03.12
申请人 JIANGSU SIMCERE PHARMACEUTICAL R&D CO., LTD.;TANG, FENG;JIN, QIU;LI, WEI;ZHU, TIAN;HU, YANG;SHAO, FENG 发明人 TANG, FENG;JIN, QIU;LI, WEI;ZHU, TIAN;HU, YANG;SHAO, FENG
分类号 C07D209/42;A61K31/404;A61P35/00 主分类号 C07D209/42
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