发明名称 PYRROLOPYRIDAZINE JAK3 INHIBITORS AND THEIR USE FOR THE TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES
摘要 <p>Disclosed are compounds of Formula (I), and pharmaceutically acceptable salts thereof. The compounds of formula (I) inhibit tyrosine kinase activity of JAK3, thereby making them useful for the treatment of inflammatory and autoimmune diseases.</p>
申请公布号 WO2012125886(A1) 申请公布日期 2012.09.20
申请号 WO2012US29334 申请日期 2012.03.16
申请人 BRISTOL-MYERS SQUIBB COMPANY;WROBLESKI, STEPHEN T.;BROWN, GREGORY D.;DOWEYKO, LIDIA M.;DUAN, JINGWU;GUO, JUNQING;HYNES, JOHN;JIANG, BIN;KEMPSON, JAMES;LIN, SHUQUN;LU, ZHONGHUI;SPERGEL, STEVEN, H.;TOKARSKI, JOHN S.;WU, HONG;YANG, BINGWEI VERA 发明人 WROBLESKI, STEPHEN T.;BROWN, GREGORY D.;DOWEYKO, LIDIA M.;DUAN, JINGWU;GUO, JUNQING;HYNES, JOHN;JIANG, BIN;KEMPSON, JAMES;LIN, SHUQUN;LU, ZHONGHUI;SPERGEL, STEVEN, H.;TOKARSKI, JOHN S.;WU, HONG;YANG, BINGWEI VERA
分类号 A61K31/5025;A61P17/00;A61P19/00;A61P29/00;A61P37/00;C07D487/04;C07D519/00 主分类号 A61K31/5025
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