发明名称 |
CRYSTALLINE FORMS OF (3R, 3AS, 6AR) - HEXAHYDROFURO [2,3-B] FURAN-3-YL (1S,2R) - (1-{4-[ (DIETHOXYPHOSPHORYL) METHOXY] PHENY1}-3-HYDROXY-4- [4-METHOXY-N- (2-METHYLPROPYL) BENZENESUL - FONAMIDO] BUTAN-2-YL) CARBAMATE |
摘要 |
The present inventions provides crystalline forms of (3R,3aS,6aR)-hexahydrofuro[2,3-b]furan-3-yl (1S,2R)-(1-{4-[(diethoxyphosphoryl)methoxy]phenyl}-3-hydroxy-4-[4-methoxy-N-(2-methylpropyl)benzenesulfonamido]butan-2-yl)carbamate, methods of preparing the crystalline forms, pharmaceutical compositions containing the crystalline forms, and therapeutic uses thereof.
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申请公布号 |
US2012232038(A1) |
申请公布日期 |
2012.09.13 |
申请号 |
US201013378250 |
申请日期 |
2010.06.17 |
申请人 |
CARRA ERNEST ANTHONY;CHIU ANNA;JERNELIUS JESPER ALEXIS;WANG FANG;GILEAD SCIENCES, INC. |
发明人 |
CARRA ERNEST ANTHONY;CHIU ANNA;JERNELIUS JESPER ALEXIS;WANG FANG |
分类号 |
A61K31/665;A61P31/18;C07F9/40 |
主分类号 |
A61K31/665 |
代理机构 |
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