发明名称 MST1 KINASE INHIBITORS AND METHODS OF THEIR USE
摘要 Compounds for the inhibition of mammalian Ste20-like kinase 1 (MST1) are disclosed, along with compositions comprising them and methods of their use in the treatment, management or prevention of an inflammatory or autoimmune diseases or disorders.
申请公布号 WO2012121992(A1) 申请公布日期 2012.09.13
申请号 WO2012US27376 申请日期 2012.03.02
申请人 LEXICON PHARMACEUTICALS, INC.;AUGERI, DAVID JOHN;BAGDANOFF, JEFFREY THOMAS;BAUGH, SIMON DAVID PETER;CARLSEN, MARIANNE;CARSON, KENNETH GORDON;GILLERAN, JOHN ANTHONY;HE, WEI;ORAVECZ, TAMAS;SALOJIN, KONSTANTIN;SUNG, LEONARD 发明人 AUGERI, DAVID JOHN;BAGDANOFF, JEFFREY THOMAS;BAUGH, SIMON DAVID PETER;CARLSEN, MARIANNE;CARSON, KENNETH GORDON;GILLERAN, JOHN ANTHONY;HE, WEI;ORAVECZ, TAMAS;SALOJIN, KONSTANTIN;SUNG, LEONARD
分类号 C07D401/04;A61K31/4418;A61K31/4725;A61K31/497;A61K31/5513;A61K31/553;A61P29/00;C07D401/14;C07D403/04;C07D405/14;C07D409/14;C07D413/04;C07D417/14;C07D471/04;C07D495/04 主分类号 C07D401/04
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