发明名称 CRYSTALLINE FORMS OF N-(TERT-BUTOXYCARBONYL)-3-METHYL-L-VALYL-(4R)-4-((7-CHLORO-4-METHOXY-1-ISOQUINOLINYL)OXY)-N-((1R,2S)-1-((CYCLOPROPYLSULFONYL)CARBAMOYL)-2-VINYLCYCLOPROPYL)-L-PROLINAMIDE
摘要 The present disclosure generally relates to crystalline forms of N-(tert-butoxycarbonyl)-3-methyl-L-valyl-(4R)-4-((7-chloro-4-methoxy-1-isoquinolinyl)oxy)-N-((1R,2S)-1-((cyclopropylsulfonyl)carbamoyl)-2-vinylcyclopropyl)-L-prolinamide. The present disclosure also generally relates to a pharmaceutical composition comprising one or more of the crystalline forms, as well of methods of using the crystalline forms in the treatment of Hepatitis C virus (HCV) and methods for obtaining such crystalline forms.
申请公布号 US2012230949(A1) 申请公布日期 2012.09.13
申请号 US201213472720 申请日期 2012.05.16
申请人 PERRONE ROBERT KEVIN;SONG ANNE I.;WANG CHENCHI;YING WILLIAM;BRISTOL-MYERS SQUIBB COMPANY 发明人 PERRONE ROBERT KEVIN;SONG ANNE I.;WANG CHENCHI;YING WILLIAM
分类号 A61K38/05;A61K38/20;A61K38/21;A61P31/14;C07D401/12 主分类号 A61K38/05
代理机构 代理人
主权项
地址