发明名称 |
PHENOXY-SUBSTITUTED PYRIMIDINES AS OPIOID RECEPTOR MODULATORS |
摘要 |
Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula I as follows: wherein R1, Y, R2, R3, and Ra are defined herein. |
申请公布号 |
EP2493863(A1) |
申请公布日期 |
2012.09.05 |
申请号 |
EP20100776483 |
申请日期 |
2010.10.28 |
申请人 |
JANSSEN PHARMACEUTICA NV |
发明人 |
COATS, STEVEN, J.;ZHANG, YUE-MEI;LIN, SHU-CHEN;LIU, LI;MISKOWSKI, TAMARA, A.;DAX, SCOTT, L.;BRESLIN, HENRY;DE CORTE, BART, L.;HE, WEI |
分类号 |
C07D239/28;A61K31/506;A61P25/04;C07D239/34;C07D401/12;C07D403/12;C07D413/12;C07D417/12 |
主分类号 |
C07D239/28 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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