发明名称 7-AMINO ALKYLIDENYL-HETEROCYCLIC QUINOLONE AND NAPHTHYRIDONE
摘要 <P>PROBLEM TO BE SOLVED: To provide new broad-spectrum antimicrobial agents, which are effective against resistant. <P>SOLUTION: The present invention relates to: compounds represented by the following formula I, wherein R is selected from hydrogen, hydroxy, and alkoxy, R<SB POS="POST">2</SB>is hydrogen, R<SB POS="POST">3</SB>and R<SB POS="POST">4</SB>are independently selected from hydrogen, halogen, amino, hydroxy, alkoxy or the like, R<SB POS="POST">5</SB>is selected from hydrogen, halogen, alkyl or the like, R<SB POS="POST">6</SB>is independently alkyl, hydroxy, alkoxy or the like; or an optical isomer, diastereomer or enantiomer thereof; and a pharmaceutically acceptable salt, hydrate, or prodrug thereof. <P>COPYRIGHT: (C)2012,JPO&INPIT
申请公布号 JP2012162529(A) 申请公布日期 2012.08.30
申请号 JP20120050624 申请日期 2012.03.07
申请人 JANSSEN PHARMACEUTICA NV 发明人 BOWERS GRANT EUGENE III;MACIELAG MARK JOSEPH;XU XIAOQING;PAGET STEVEN DAVID;WEIDNER-WELLS MICHELE ANN
分类号 C07D401/04;A61K31/435;A61K31/4523;A61K31/47;A61K31/4709;A61K31/4745;A61K31/519;A61K31/5365;A61P31/04;C07D403/04;C07D471/02;C07D471/04;C07D487/04;C07D498/06 主分类号 C07D401/04
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