发明名称 SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE
摘要 This invention comprises the novel compounds of formula (I) wherein R1, R2, R3, X and Y have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
申请公布号 US2012220615(A1) 申请公布日期 2012.08.30
申请号 US201213447636 申请日期 2012.04.16
申请人 VERDONCK MARC GUSTAAF CELINE;ANGIBAUD PATRICK RENE;ROUX BRUNO;PILATTE ISABELLE NOELLE CONSTANCE;TEN HOLTE PETER;ARTS JANINE;VAN EMELEN KRISTOF 发明人 VERDONCK MARC GUSTAAF CELINE;ANGIBAUD PATRICK RENE;ROUX BRUNO;PILATTE ISABELLE NOELLE CONSTANCE;TEN HOLTE PETER;ARTS JANINE;VAN EMELEN KRISTOF
分类号 C07D401/14;A61K31/506;A61P35/04;C07D405/14;C07D409/14;C07D491/04 主分类号 C07D401/14
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