| 摘要 |
FIELD: chemistry. ^ SUBSTANCE: invention relates to novel phenyl-pyrimidinyl-amino derivatives of formula (I), as well as agriculturally acceptable salts thereof, having fungicidal activity, a composition and a method of controlling phytopathogenic fungi of agricultural crops. In formula (I) Q1 independently represents a halogen atom, C1-C8alkyl, C1-C8halogenalkyl, having 1-5 halogen atoms, C2-C8alkenyl, C2-C8alkenyloxy, C1-C8alkoxy, C1-C8halogenalkoxy, having 1-5 halogen atoms, C1-C8alkylcarbonyl, C1-C8alkylcarbonylamino, C1-C8halogenalkylcarbonylamino, having 1-5 halogen atoms, C1-C8alkylsulphanyl, C1-C8halogenalkylsulphanyl, having 1-5 halogen atoms, C1-C8alkylsulphonyl, C1-C8halogenalkylsulphonyl, having 1-5 halogen atoms, C1-C8alkoxyalkyl, C1-C8halogenalkoxyalkyl, having 1-5 halogen atoms; p= 0, 1, 2, 3, 4 or 5; Ra represents a hydrogen atom, C1-C8alkylcarbonyl; Rb and Rc independently represent a hydrogen atom, L1 represents an unsubstituted pyridin-3-yl or pyridin-4-yl; where the group Q2-L2-CY lies in the alpha-position relative the nitrogen ring atom; Y represents O, S, NRd; L2 represents a direct bond, O, NRg; Q2 represents a hydrogen atom, substituted or unsubstitured C1-C8alkyl, substituted or unsubstituted C3-C8cycloalkyl; C2-C8alkenyl, (2-oxopyrrolidin-1-yl)-C1-C8alkyl, (2-oxoazepan-1-yl)-C1-C8alkyl, (2-oxopyrrolidin-1-yl)-C1-C8halogenalkyl, having 1 -5 halogen atoms; (2-oxoazepan-1-yl)-C1-C8halogenalkyl, having 1-5 halogen atoms; where the substitutes are selected from a group consisting of a halogen atom, a hydroxy group, di C1-C8alkylamino, C1-C8alkoxy; or L2 and Q2 together can form a substituted or unsubstituted 4-, 5-, 6- or 7-member heterocycle, containing up to 4 heteroatoms, selected from a list consisting of N, O, S, where the substitutes are independently selected from a group consisting of a halogen atom, a hydroxy group, di C1-C8alkylamino, C1-C8alkoxy; Rd represents a hydroxy group, C1-C8alkoxy, C2-C8alkenyloxy; Rg represents a hydrogen atom, C1-C8alkyl, C3-C6cycloalkyl, C2-C8alkenyl or C1-C8alkoxy. ^ EFFECT: obtaining novel phenyl-pyrimidinyl-amino derivatives of formula (I), as well as agriculturally acceptable salts thereof, having fungicidal activity. ^ 11 cl, 11 tbl, 5 ex |
