发明名称 |
SPIRO-CONDENSED CYCLOHEXANE DERIVATIVES AS HSL INHIBITORS USEFUL FOR THE TREATMENT OF DIABETES |
摘要 |
<p>The present invention relates to compounds of formula (I) as well as pharmaceutically acceptable salts thereof. The are useful as HSL inhibitors and may, for example, be used in treatment of diabetes, metabolic syndrome, dyslipidemia, atherosclerosis, and obesity.</p> |
申请公布号 |
EP2488493(A1) |
申请公布日期 |
2012.08.22 |
申请号 |
EP20100770764 |
申请日期 |
2010.10.12 |
申请人 |
F.HOFFMANN-LA ROCHE AG |
发明人 |
ACKERMANN, JEAN;BRUGGER, STEPHAN;CONTE, AURELIA;HUNZIKER, DANIEL;NEIDHART, WERNER;NETTEKOVEN, MATTHIAS;SCHULZ-GASCH, TANJA;WERTHEIMER, STANLEY |
分类号 |
C07D209/54;A61K31/403;A61P3/00;C07D401/06;C07D401/12;C07D403/12;C07D405/04;C07D405/12;C07D409/12;C07D413/12 |
主分类号 |
C07D209/54 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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