发明名称 PROCESS FOR THE PREPARATION OF ATOVAQUONE
摘要 Disclosed herein is novel process for preparation of atovaquone, which process includes reacting1H-2-benzopyran-1,4(3H)-dione with 4-(4-chlorophenyl)cyclohexanecarbaldehyde. The invention further discloses novel intermediates useful in the preparation of atovaquone.
申请公布号 WO2012080243(A3) 申请公布日期 2012.08.16
申请号 WO2011EP72600 申请日期 2011.12.13
申请人 GLAXO GROUP LIMITED;DWYER, ANDREW NEIL;GORDON, ANDREW;URQUHART, MICHAEL 发明人 DWYER, ANDREW NEIL;GORDON, ANDREW;URQUHART, MICHAEL
分类号 C07C46/00;C07C50/32;C07C69/78;C07D307/89;C07D311/76 主分类号 C07C46/00
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