发明名称 BAFF BINDING INHIBITOR HAVING 4-(2-BENZYLIDENE HYDRAZINYL)-2-PHENYLPYRIMIDINE DERIVATIVE AS ACTIVE INGREDIENT
摘要 <P>PROBLEM TO BE SOLVED: To provide a drug which inhibits the BAFF binding to a BR3 receptor and has excellent preventing and treating effects on autoimmune diseases, acquired immunodeficiency syndrome, and non-Hodgkin lymphoma. <P>SOLUTION: The BAFF binding inhibitor to a BR3 receptor includes a compound represented by formula (1) (wherein R<SP POS="POST">1</SP>is a 1-10C alkyl group; and R<SP POS="POST">2</SP>, R<SP POS="POST">3</SP>, R<SP POS="POST">4</SP>, and R<SP POS="POST">5</SP>may be the same as or different from one another and are each hydrogen or a hydroxyl group), a salt thereof or a solvate thereof as an active ingredient. <P>COPYRIGHT: (C)2012,JPO&INPIT
申请公布号 JP2012144442(A) 申请公布日期 2012.08.02
申请号 JP20110001505 申请日期 2011.01.06
申请人 TAKEUCHI TSUTOMU;NATIONAL INSTITUTE OF ADVANCED INDUSTRIAL SCIENCE& TECHNOLOGY;KOWA CO 发明人 TAKEUCHI TSUTOMU;YOSHIMOTO KEIKO;HIROKAWA TAKATSUGU;YAMADA HAJIME;OKUDA AYUMI;ITO NAOHIRO;SUGANO TOMOHIRO
分类号 A61K31/505;A61P17/00;A61P19/02;A61P25/00;A61P29/00;A61P35/00;A61P37/02;A61P43/00;C07D239/42 主分类号 A61K31/505
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