发明名称 |
2-HYDROXYMETHYL-3,4,5-TRIHYDROXY-1-(4-PENTLYOXYBENZYL) PIPERIDINE AS GLUCOSYLCERAMIDE SYNTHASE (GCS) |
摘要 |
The compound 3,4,5-piperidinetriol, 2-(hydroxymethyl)-1-[(4-(pentyloxy)phenyl)methyl]-, (2S,3S,4R,5S), or a pharmaceutically acceptable salt or prodrug thereof, is useful as an inhibitor of glucosylceramide synthase.
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申请公布号 |
CA2528322(C) |
申请公布日期 |
2012.07.31 |
申请号 |
CA20042528322 |
申请日期 |
2004.06.09 |
申请人 |
ACTELION PHARMACEUTICALS LTD |
发明人 |
ORCHARD, MICHAEL GLEN;SCOPES, DAVID IAN CARTER |
分类号 |
C07D211/46;A61K31/445;A61P3/10;A61P35/00 |
主分类号 |
C07D211/46 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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