发明名称 AMINOPYRIMIDINES AS SYK INHIBITORS
摘要 <p>The present invention provides novel pyrimidine amines of formula (I) which are potent inhibitors of spleen tyrosine kinase, and are useful in the treatment and prevention of diseases mediated by said enzyme, such as asthma, COPD and rheumatoid arthritis.</p>
申请公布号 SG181803(A1) 申请公布日期 2012.07.30
申请号 SG20120045118 申请日期 2010.12.15
申请人 MERCK SHARP & DOHME CORP.;MERCK CANADA INC. 发明人 ALTMAN, MICHAEL, D.;ANDRESEN, BRIAN, M.;ARRINGTON, KENNETH, L.;CHILDERS, KALEEN, KONRAD;DI FRANCESCO, MARIA, EMILIA;DONOFRIO, ANTHONY;ELLIS, JOHN, MICHAEL;FISCHER, CHRISTIAN;GUERIN, DAVID, JOSEPH;HAIDLE, ANDREW, M.;KATTAR, SOLOMON;KNOWLES, SANDRA, LEE;LI, CHAOMIN;LIM, JONGWON;MACHACEK, MICHELLE, R.;NORTHRUP, ALAN, B.;O'BOYLE, BRENDAN, M.;OTTE, RYAN, D.;PETROCCHI, ALESSIA;REUTERSHAN, MICHAEL, H.;ROMEO, ERIC;SIU, TONY;TAOKA, BRANDON, M.;TROTTER, B., WESLEY;ZHOU, HUA;BURCH, JASON;COTE, BERNARD;DUPONT-GAUDET, KRISTINA;FOURNIER, JEAN-FRANCOIS;GAUTHIER, JACQUES, YVES;GUAY, DANIEL;ROBICHAUD, JOEL, S.
分类号 主分类号
代理机构 代理人
主权项
地址