发明名称 |
INDOLYL-PIPERIDINYL BENZYLAMINES AS BETA-TRYPTASE INHIBITORS |
摘要 |
<p>The present invention discloses and claims a series of substituted indolyl-piperidinyl benzylamines of formula (I), wherein R1, R2 and R3 are as described herein. More specifically, the compounds of this invention are inhibitors ofβ-tryptase and are, therefore, useful as pharmaceutical agents. Additionally, this invention also discloses methods of preparation of substituted indolyl-piperidinyl benzylamines. In one of the embodiments, there is provided the compounds of formula (I) wherein R3 is (II).</p> |
申请公布号 |
SG181504(A1) |
申请公布日期 |
2012.07.30 |
申请号 |
SG20120040994 |
申请日期 |
2010.12.21 |
申请人 |
SANOFI |
发明人 |
CHOI-SLEDESKI, YONG MI;LIANG, GUYAN;NIEDUZAK, THADDEUS R.;POLI, GREGORY B.;SHUM, PATRICK WAI-KWOK;STOKLOSA, GREGORY T.;ZHAO, ZHICHENG |
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