发明名称 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-B]PYRIDINES AND PYRROLO[2,3- B]PYRIMIDINES AS JANUS KINASE INHIBITORS |
摘要 |
The present invention provides heteroaryl substituted pyrrolo[2,3-b]pyridines (I) and heteroaryl substituted pyrrolo[2,3-b]pyrimidines that modulate the activity of Janus kinases and are useful in the treatment of diseases related to activity of Janus kinases including, for example, immune-related diseases, skin disorders, myeloid proliferative disorders, cancer, and other diseases. |
申请公布号 |
HK1124840(A1) |
申请公布日期 |
2012.07.27 |
申请号 |
HK20090102199 |
申请日期 |
2009.03.06 |
申请人 |
INCYTE CORPORATION |
发明人 |
RODGERS, JAMES D.;SHEPARD, STACEY;MADUSKUIE, THOMAS P.;WANG, HAISHENG;FALAHATPISHEH, NIKOO;RAFALSKI, MARIA;ARVANITIS, ARGYRIOS G.;STORACE, LOUIS;JALLURI, RAVI KUMAR;FRIDMAN, JORDAN S.;VADDI, KRISHNA |
分类号 |
A61K;A61P;C07D |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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