The present invention provides a preparation with improved disintegration property, a preparation showing improved bioavailability of a medicament, production methods thereof and the like. A rapidly disintegrating preparation comprising granules comprising a medicament coated with a coating layer containing sugar or sugar alcohol; and a disintegrant. A production method of a rapidly disintegrating preparation including a step of producing granules comprising a medicament, a step of forming a coating layer containing sugar or sugar alcohol on the obtained granules and a step of mixing the coated granules with a disintegrant and molding the mixture.
申请公布号
WO2012099260(A1)
申请公布日期
2012.07.26
申请号
WO2012JP51279
申请日期
2012.01.16
申请人
TAKEDA PHARMACEUTICAL COMPANY LIMITED;TANOUE, YUTAKA;MATSUURA, TETSUYA;YAMAGATA, YUTAKA;NAGAHARA, NAOKI