发明名称 PROCESS FOR THE PREPARATION OF N- [2 - (7 -METHOXY - 1 - NAPHTHYL) - ETHYL] ACETAMIDE AND NEW CRYSTALLINE FORM
摘要 A novel process for the preparation of N-[2-(7-methoxy-1-naphthyl)ethyl]acetamide, also known as agomelatine, Compound (I), from 7-methoxy-tetralone as starting material, and to a new crystalline form X of agomelatine.
申请公布号 WO2011154140(A3) 申请公布日期 2012.07.26
申请号 WO2011EP02834 申请日期 2011.06.09
申请人 GADOR S.A.;CONICET -CONSEJO NAC. DE INVESTIGACIONES CIENTIFICAS Y TECNICAS;TOMBARI, DORA, GRACIELA;MANGONE, CONSTANZA, PIA;GARCIA, MARIA, BEATRIZ;VECCHIOLI, ADRIANA;LABRIOLA, RAFAEL, ALBERTO;BURTON, GERARDO;RUSTOY, EDUARDO, MIGUEL 发明人 TOMBARI, DORA, GRACIELA;MANGONE, CONSTANZA, PIA;GARCIA, MARIA, BEATRIZ;VECCHIOLI, ADRIANA;LABRIOLA, RAFAEL, ALBERTO;BURTON, GERARDO;RUSTOY, EDUARDO, MIGUEL
分类号 C07C217/74;C07C233/18;C07C255/37 主分类号 C07C217/74
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