Process for the preparation of asenapine and intermediate products used in said process
摘要
The invention relates to a novel process for the preparation of asenapine, i.e. trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, as well as to novel intermediate products for use in said process.
申请公布号
US8227623(B2)
申请公布日期
2012.07.24
申请号
US20100785805
申请日期
2010.05.24
申请人
KEMPERMAN GERARDUS JOHANNES;STUK TIMOTHY LEE;VAN DER LINDEN JACOBUS JOHANNES MARIA;MSD OSS B.V.
发明人
KEMPERMAN GERARDUS JOHANNES;STUK TIMOTHY LEE;VAN DER LINDEN JACOBUS JOHANNES MARIA