发明名称 Process for the preparation of asenapine and intermediate products used in said process
摘要 The invention relates to a novel process for the preparation of asenapine, i.e. trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, as well as to novel intermediate products for use in said process.
申请公布号 US8227623(B2) 申请公布日期 2012.07.24
申请号 US20100785805 申请日期 2010.05.24
申请人 KEMPERMAN GERARDUS JOHANNES;STUK TIMOTHY LEE;VAN DER LINDEN JACOBUS JOHANNES MARIA;MSD OSS B.V. 发明人 KEMPERMAN GERARDUS JOHANNES;STUK TIMOTHY LEE;VAN DER LINDEN JACOBUS JOHANNES MARIA
分类号 C07D207/04 主分类号 C07D207/04
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