发明名称 SOLID FORMS OF GYRASE INHIBITOR (R)-1-ETHYL-3-[6-FLUORO-5-[2-(1-HYDROXY-1-METHYL-ETHYL)PYRIMIDIN-5-YL]-7-(TETRAHYDROFURAN-2-YL)-1H-BENZIMIDAZOL-2-YL]UREA
摘要 The present application is directed to solid forms of compounds of formula I: and pharmaceutically acceptable salts thereof, that inhibit bacterial gyrase and/or Topo IV and pharmaceutical compositions comprising said compounds and salts. These compounds and salts are useful in treating bacterial infections.
申请公布号 US2012184564(A1) 申请公布日期 2012.07.19
申请号 US201213349984 申请日期 2012.01.13
申请人 SHANNON DEAN;LUISI BRIAN;KRAWIEC MARIUSZ;KULDIPKUMAR ANUJ K.;VERTEX PHARMACEUTICALS INCORPORATED 发明人 SHANNON DEAN;LUISI BRIAN;KRAWIEC MARIUSZ;KULDIPKUMAR ANUJ K.
分类号 A61K31/506;A61P31/04;C07D405/14 主分类号 A61K31/506
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