发明名称 |
METHOD OF PREPARING POLYMORPHIC PURE FORM A OF BAZEDOXIFENE ACETATE |
摘要 |
The present invention provides a reliable process for the preparation of polymorphic pure form A of Bazedoxifene x acetate. In addition, the present invention relates to a process of wet granulation of polymorphic pure form A of Bazedoxifene x acetate. The present invention also relates to pharmaceutical compositions comprising polymorphic pure form A of Bazedoxifene x acetate as well as to the use of cyclic ethers for the preparation of such pharmaceutical composition. |
申请公布号 |
WO2012089593(A1) |
申请公布日期 |
2012.07.05 |
申请号 |
WO2011EP73669 |
申请日期 |
2011.12.21 |
申请人 |
SANDOZ AG;PICHLER, ARTHUR;HOTTER, ANDREAS;LANGES, CHRISTOPH |
发明人 |
PICHLER, ARTHUR;HOTTER, ANDREAS;LANGES, CHRISTOPH |
分类号 |
C07D209/12;A61K31/404;A61K31/55;A61P19/10 |
主分类号 |
C07D209/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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