发明名称 Process for preparing rosuvastatin calcium
摘要 The present invention relates to an improved process for preparing (2E)-3-[4-(4-fluorophenyl)-6-iso-propyl-2-(N-methyl-N-methylsulfonylamino)pyrimidin-5-yl]-propenal of Formula I which is an intermediate useful in the preparation of bis[(E)-7-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino]pyrimidin-5-yl](3R,5S)-3,5-dihydroxyhept-6-enoicacid]calcium salt of Formula II.
申请公布号 US8212034(B2) 申请公布日期 2012.07.03
申请号 US20070448270 申请日期 2007.12.11
申请人 DANDALA RAMESH;MALLELA SAMBHU PRASAD SARMA;NANDI SUKUMAR;NANGI GANGADHAR BHIMA SHANKAR;BURIDIPADU SUNIL KUMAR;MEENAKSHISUNDERAM SIVAKUMARAN;AUROBINDO PHARMA LTD. 发明人 DANDALA RAMESH;MALLELA SAMBHU PRASAD SARMA;NANDI SUKUMAR;NANGI GANGADHAR BHIMA SHANKAR;BURIDIPADU SUNIL KUMAR;MEENAKSHISUNDERAM SIVAKUMARAN
分类号 C07D239/42 主分类号 C07D239/42
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