发明名称 SPIROPIPERIDINES FOR USE AS TRYPTASE INHIBITORS
摘要 The present invention is directed to a compound of Formula (I): or a form thereof, wherein X1, X2, X3, X4, R1, R2 and R3 are as defined herein, useful as tryptase inhibitors.
申请公布号 US2012165327(A1) 申请公布日期 2012.06.28
申请号 US201213409559 申请日期 2012.03.01
申请人 COSTANZO MICHAEL J.;YABUT STEPHEN C.;TOUNGE BRETT;MARYANOFF BRUCE E.;ZHANG HAN-CHENG 发明人 COSTANZO MICHAEL J.;YABUT STEPHEN C.;TOUNGE BRETT;MARYANOFF BRUCE E.;ZHANG HAN-CHENG
分类号 A61K31/438;A61K31/444;A61K31/506;A61K31/5377;A61P1/00;A61P1/04;A61P1/16;A61P9/00;A61P9/08;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/12;A61P17/00;A61P17/02;A61P17/04;A61P17/06;A61P19/02;A61P27/02;A61P29/00;A61P37/00;A61P37/08;C07D405/06;C07D471/10;C07D491/107;C07D495/04;C07D495/10 主分类号 A61K31/438
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