发明名称 |
SPIROPIPERIDINES FOR USE AS TRYPTASE INHIBITORS |
摘要 |
The present invention is directed to a compound of Formula (I): or a form thereof, wherein X1, X2, X3, X4, R1, R2 and R3 are as defined herein, useful as tryptase inhibitors. |
申请公布号 |
US2012165327(A1) |
申请公布日期 |
2012.06.28 |
申请号 |
US201213409559 |
申请日期 |
2012.03.01 |
申请人 |
COSTANZO MICHAEL J.;YABUT STEPHEN C.;TOUNGE BRETT;MARYANOFF BRUCE E.;ZHANG HAN-CHENG |
发明人 |
COSTANZO MICHAEL J.;YABUT STEPHEN C.;TOUNGE BRETT;MARYANOFF BRUCE E.;ZHANG HAN-CHENG |
分类号 |
A61K31/438;A61K31/444;A61K31/506;A61K31/5377;A61P1/00;A61P1/04;A61P1/16;A61P9/00;A61P9/08;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/12;A61P17/00;A61P17/02;A61P17/04;A61P17/06;A61P19/02;A61P27/02;A61P29/00;A61P37/00;A61P37/08;C07D405/06;C07D471/10;C07D491/107;C07D495/04;C07D495/10 |
主分类号 |
A61K31/438 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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