发明名称 |
PREPARATION OF PROTECTED ALPHA-KETO BETA-AMINO ESTERS AND AMIDES |
摘要 |
The invention provides &bgr;-sulfonamide α-keto esters and amides in which the α-keto is protected as a 1,3-dithiolane derivative. Also provided are methods for preparing such esters and amides and for incorporating them into peptides. |
申请公布号 |
ZA201100226(B) |
申请公布日期 |
2012.06.27 |
申请号 |
ZA20110000226 |
申请日期 |
2011.01.07 |
申请人 |
VERTEX PHARMACEUTICALS INCORPORATED |
发明人 |
NUGENT WILLIAM A;LOOKER ADAM R;FORSLUND RAYMOND E;MARTINOT THEODORE A;HARRISON CRISTIAN L;IBRAHIM SHEREE |
分类号 |
C07D |
主分类号 |
C07D |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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