发明名称 PREPARATION OF PROTECTED ALPHA-KETO BETA-AMINO ESTERS AND AMIDES
摘要 The invention provides &bgr;-sulfonamide α-keto esters and amides in which the α-keto is protected as a 1,3-dithiolane derivative. Also provided are methods for preparing such esters and amides and for incorporating them into peptides.
申请公布号 ZA201100226(B) 申请公布日期 2012.06.27
申请号 ZA20110000226 申请日期 2011.01.07
申请人 VERTEX PHARMACEUTICALS INCORPORATED 发明人 NUGENT WILLIAM A;LOOKER ADAM R;FORSLUND RAYMOND E;MARTINOT THEODORE A;HARRISON CRISTIAN L;IBRAHIM SHEREE
分类号 C07D 主分类号 C07D
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