发明名称 Development of molecular imaging probes for carbonic anhydrase-IX using click chemistry
摘要 <p>The present application discloses methods for identifying inhibitors with high binding-affinity for the carbonic anhydrase-IX (CA-IX) enzyme using click chemistry and uses the candidates thereof as positron emission tomography (PET) imaging agents.</p>
申请公布号 EP2468734(A1) 申请公布日期 2012.06.27
申请号 EP20120157766 申请日期 2008.04.07
申请人 SIEMENS MEDICAL SOLUTIONS USA, INC. 发明人 KOLB, HARTMUTH;CHEN, GANG;PADGETT, HENRY;KARIMI, FARHAD;SCOTT, PETER;GAO, ZHIYONG;LIANG, QIANWA;COLLIER, THOMAS LEE;ZHAO, TIEMING;XIA, CHUNFANG;WALSH, JOSEPH;KASI, DHANALAKSHMI;MOCHARLA, VANI;WANG, BING;GANGADHARMATH, UMESH;DUCLOS, BRIAN;CHEN, KAI;ZHANG, WEI
分类号 C07D249/04;A61K31/4192;A61P35/00;C07D249/06;C07D401/04;C07D401/12;C07D403/04;C07D403/12;C07D405/04;C07D405/12;C07D409/12;C07D417/04;C07D417/12;C07D417/14;G01N33/532 主分类号 C07D249/04
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