发明名称 |
FUSED DIHYDROPYRANS AS GPR119 MODULATORS FOR THE TREATMENT OF DIABETES, OBESITY AND RELATED DISEASES |
摘要 |
The present invention relates to compounds of general formula (I), wherein the groups R1, LP, LQ, X1, X2, X3, Ar and n are as defined in the application, which have valuable pharmacological properties, and in particular bind to the GPR119 receptor and modulate its activity. |
申请公布号 |
WO2012080476(A1) |
申请公布日期 |
2012.06.21 |
申请号 |
WO2011EP73067 |
申请日期 |
2011.12.16 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH;HIMMELSBACH, FRANK;ECKHARDT, MATTHIAS;HEINE, NIKLAS;LANGKOPF, ELKE;NOSSE, BERND |
发明人 |
HIMMELSBACH, FRANK;ECKHARDT, MATTHIAS;HEINE, NIKLAS;LANGKOPF, ELKE;NOSSE, BERND |
分类号 |
C07D407/04;A61K31/4525;A61K31/4545;A61K31/496;A61K31/497;A61K31/4985;A61K31/501;A61K31/519;A61K31/5377;A61P3/10;C07D407/14;C07D409/14;C07D413/14;C07D417/14;C07D491/048 |
主分类号 |
C07D407/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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