发明名称 FUSED DIHYDROPYRANS AS GPR119 MODULATORS FOR THE TREATMENT OF DIABETES, OBESITY AND RELATED DISEASES
摘要 The present invention relates to compounds of general formula (I), wherein the groups R1, LP, LQ, X1, X2, X3, Ar and n are as defined in the application, which have valuable pharmacological properties, and in particular bind to the GPR119 receptor and modulate its activity.
申请公布号 WO2012080476(A1) 申请公布日期 2012.06.21
申请号 WO2011EP73067 申请日期 2011.12.16
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH;HIMMELSBACH, FRANK;ECKHARDT, MATTHIAS;HEINE, NIKLAS;LANGKOPF, ELKE;NOSSE, BERND 发明人 HIMMELSBACH, FRANK;ECKHARDT, MATTHIAS;HEINE, NIKLAS;LANGKOPF, ELKE;NOSSE, BERND
分类号 C07D407/04;A61K31/4525;A61K31/4545;A61K31/496;A61K31/497;A61K31/4985;A61K31/501;A61K31/519;A61K31/5377;A61P3/10;C07D407/14;C07D409/14;C07D413/14;C07D417/14;C07D491/048 主分类号 C07D407/04
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