发明名称 SUBSTITUTED N-(1H-INDAZOL-4-YL)IMIDAZO[1,2-a]PYRIDINE-3-CARBOXAMIDE COMPOUNDS AS TYPE III RECEPTOR TYROSINE KINASE INHIBITORS
摘要 Compounds of Formula I: and pharmaceutically acceptable salts thereof in which R1, R2, R3, R4, R5 and R6 have the meanings given in the specification, are inhibitors of cFMS and are useful in the treatment of fibrosis, bone-related diseases, cancer, autoimmune disorders, inflammatory diseases, cardiovascular diseases, pain and burns in a mammal.
申请公布号 WO2012082689(A1) 申请公布日期 2012.06.21
申请号 WO2011US64549 申请日期 2011.12.13
申请人 ARRAY BIOPHARMA INC.;BOYS, MARK LAURENCE;DELISLE, ROBERT KIRK;HICKEN, ERIK JAMES;KENNEDY, APRIL L.;MARESKA, DAVID A.;MARMSATER, FREDRIK P.;MUNSON, MARK C.;NEWHOUSE, BRAD;RAST, BRYSON;RIZZI, JAMES P.;RODRIGUEZ, MARTHA E.;TOPALOV, GEORGE T.;ZHAO, QIAN 发明人 BOYS, MARK LAURENCE;DELISLE, ROBERT KIRK;HICKEN, ERIK JAMES;KENNEDY, APRIL L.;MARESKA, DAVID A.;MARMSATER, FREDRIK P.;MUNSON, MARK C.;NEWHOUSE, BRAD;RAST, BRYSON;RIZZI, JAMES P.;RODRIGUEZ, MARTHA E.;TOPALOV, GEORGE T.;ZHAO, QIAN
分类号 C07D471/04;A61K31/437;A61P35/00 主分类号 C07D471/04
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