发明名称 SUBSTITUTED AMINOPROPENYL PIPERIDINE OR MORPHOLINE DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE
摘要 This invention comprises the novel compounds of formula (I) wherein R1, R2, R3, R4, X and Y have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
申请公布号 US2012157456(A1) 申请公布日期 2012.06.21
申请号 US201113302930 申请日期 2011.11.22
申请人 ANGIBAUD PATRICK RENE;MARCONNET-DECRANE LAURENCE FRANCOISE BERNADETTE;VAN BRANDT SVEN FRANCISCUS ANNA;PILATTE ISABELLE NOELLE CONSTANCE;JANSSEN PHARMACEUTICA N.V. 发明人 ANGIBAUD PATRICK RENE;MARCONNET-DECRANE LAURENCE FRANCOISE BERNADETTE;VAN BRANDT SVEN FRANCISCUS ANNA;PILATTE ISABELLE NOELLE CONSTANCE
分类号 A61K31/5377;A61K31/506;A61P35/00;C07D401/04;C07D413/04 主分类号 A61K31/5377
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