发明名称 4-OXO-1H-QUINOLINE-3-CARBOXAMIDES AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
摘要 <p>The present invention relates to 4-oxo-1H-quinoline-3-carboxamides as modulators of ATP-Binding Cassette ("ABC") transporters or fragments thereof, including Cystic Fibrosis Transmembrane Conductance Regulator, compositions thereof, and methods therewith. The present invention also relates to methods of treating ABC transporter mediated diseases using such modulators.</p>
申请公布号 WO2011072241(A9) 申请公布日期 2012.06.14
申请号 WO2010US59920 申请日期 2010.12.10
申请人 VERTEX PHARMACEUTICALS INCORPORATED;SHETH, URVI;FANNING, LEV T.D.;NUMA, MEHDI;BINCH, HAYLEY;HURLEY, DENNIS, JAMES;ZHOU, JINGLAN;HADIDA RUAH, SARA, S.;HAZLEWOOD, ANNA, R.;SILINA, ALINA;VAIRAGOUNDAR, RAJENDRAN;VAN GOOR, FREDRICK, F.;GROOTENHUIS, PETER, DIEDERIK JAN;BOTFIELD, MARTYN, C. 发明人 SHETH, URVI;FANNING, LEV T.D.;NUMA, MEHDI;BINCH, HAYLEY;HURLEY, DENNIS, JAMES;ZHOU, JINGLAN;HADIDA RUAH, SARA, S.;HAZLEWOOD, ANNA, R.;SILINA, ALINA;VAIRAGOUNDAR, RAJENDRAN;VAN GOOR, FREDRICK, F.;GROOTENHUIS, PETER, DIEDERIK JAN;BOTFIELD, MARTYN, C.
分类号 C07D215/56;A61K31/4709;A61P11/00;C07D401/12;C07D405/12;C07D409/12;C07D413/12;C07D417/12;C07D471/08 主分类号 C07D215/56
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