发明名称 |
HETEROARYL SUBSTITUTED ARYLINDENOPYRIMIDINES AND THEIR USE AS HIGHLY SELECTIVE ADENOSINE A2A RECEPTOR ANTAGONISTS. |
摘要 |
<p>This invention relates to a novel arylindenopyrimidine, A, and its therapeutic and prophylactic uses. Disorders treated and/or prevented include Parkinson's Disease. Formula (I) wherein X, R2, R3, and R4 are as defined in the specification.</p> |
申请公布号 |
MX2012005004(A) |
申请公布日期 |
2012.06.12 |
申请号 |
MX20120005004 |
申请日期 |
2010.10.21 |
申请人 |
JANSSEN PHARMACEUTICA NV.* |
发明人 |
WANG, AIHUA;JACKSON, PAUL F.;POWELL, MARCK;SHOOK, BRIAN CRISTOPHER |
分类号 |
C07D401/04;A61K31/519;A61P25/00;A61P25/16;A61P25/22;A61P25/24;A61P25/28;A61P25/30;C07D409/04;C07D417/04 |
主分类号 |
C07D401/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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