发明名称 Salt forms of 4-(4-Methylpiperazin-1-ylmethyl)-N-[4-methyl-3-(4-pyridin-3-yl) pyrimidin-2-ylamino)phenyl]-benzamide
摘要 The present invention relates to acid addition salts of 4-[(4-methyl-1-piperazinyl)methyl]-N-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-benzamide, which are selected from the group consisting of a tartrate salt, such as a (D)(−) tartrate salt or a (L)(+) tartrate salt, a hydrochloride salt, a citrate salt, a malate salt, a fumarate salt, a succinate salt, a benzoate salt, a benzenesulfonate salt, a pamoate salt, a formate salt, a malonate salt, a 1,5-naphthalenedisulfonate salt, a salicylate salt, a cyclohexanesulfamate salt, a lactate salt, a mandelate salt, aq glutarate salt, an adipate salt, a squarate salt, a vanillate salt, an oxaloacetate salt, an ascorbate salt and a sulfate salt.
申请公布号 US2012142697(A1) 申请公布日期 2012.06.07
申请号 US201213368811 申请日期 2012.02.08
申请人 BUERGER HANS MICHAEL;MANLEY PAUL WILLIAM;MUTZ MICHAEL 发明人 BUERGER HANS MICHAEL;MANLEY PAUL WILLIAM;MUTZ MICHAEL
分类号 A61K31/506;A61P35/00;A61P35/02;C07D401/04;C07D403/14 主分类号 A61K31/506
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