发明名称 INTERMEDIATE COMPOUNDS AND PROCESSES FOR THE PREPARATION OF QUINOLINE DERIVATIVES SUCH AS LAQUINIMOD SODIUM
摘要 The present invention relates to processes for the preparation of quinoline-3 -carboxamide derivatives, such as sodium 5-chloro-3-(ethylphenylcarbamoyl)-l-methyl-2- oxo-l,2-dihydroquinolin-4-olate (Laquinimod sodium). The present invention further relates to intermediates formed in such processes.
申请公布号 WO2012070051(A1) 申请公布日期 2012.05.31
申请号 WO2011IL50030 申请日期 2011.11.28
申请人 MAPI PHARMA LTD.;MAROM, EHUD;MIZHIRITSKII, MICHAEL;RUBNOV, SHAI 发明人 MAROM, EHUD;MIZHIRITSKII, MICHAEL;RUBNOV, SHAI
分类号 A01N43/42;A61K31/47 主分类号 A01N43/42
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