发明名称 COCRYSTAL OF C-GLYCOSIDE DERIVATIVE AND L-PROLINE
摘要 A cocrystal of (1S)-1,5-anhydro-1-[3-(1-benzothien-2--ylmethyl)-4-fluorophenyl]-D-glucitol and L-proline. It is a cocrystal of known compound A, which has a constant quality, is superior in storage stability, has no moisture absorptivity, and is suitable as a crystal of a drug substance used for preparing pharmaceuticals.
申请公布号 CA2649022(C) 申请公布日期 2012.05.29
申请号 CA20072649022 申请日期 2007.04.04
申请人 ASTELLAS PHARMA INC.;KOTOBUKI PHARMACEUTICAL CO., LTD. 发明人 IMAMURA, MASAKAZU;NAKANISHI, KEITA;SHIRAKI, RYOTA;ONDA, KENICHI;SASUGA, DAISUKE;YUDA, MASAMICHI
分类号 C07D407/10;A61K31/381;A61P3/10 主分类号 C07D407/10
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