发明名称 |
COCRYSTAL OF C-GLYCOSIDE DERIVATIVE AND L-PROLINE |
摘要 |
A cocrystal of (1S)-1,5-anhydro-1-[3-(1-benzothien-2--ylmethyl)-4-fluorophenyl]-D-glucitol and L-proline. It is a cocrystal of known compound A, which has a constant quality, is superior in storage stability, has no moisture absorptivity, and is suitable as a crystal of a drug substance used for preparing pharmaceuticals.
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申请公布号 |
CA2649022(C) |
申请公布日期 |
2012.05.29 |
申请号 |
CA20072649022 |
申请日期 |
2007.04.04 |
申请人 |
ASTELLAS PHARMA INC.;KOTOBUKI PHARMACEUTICAL CO., LTD. |
发明人 |
IMAMURA, MASAKAZU;NAKANISHI, KEITA;SHIRAKI, RYOTA;ONDA, KENICHI;SASUGA, DAISUKE;YUDA, MASAMICHI |
分类号 |
C07D407/10;A61K31/381;A61P3/10 |
主分类号 |
C07D407/10 |
代理机构 |
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代理人 |
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地址 |
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