发明名称 SALTS OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE
摘要 Disclosed is a salt selected from: (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile maleic acid salt; (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile sulfuric acid salt; and (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile phosphoric acid salt. The compounds are used to treat diseases associated with the Janus Kinase (JAK) activity such as immune-related diseases, skin disorders, myeloid proliferative disorders, cancers and the like.
申请公布号 NZ581803(A) 申请公布日期 2012.05.25
申请号 NZ20080581803 申请日期 2008.06.12
申请人 INCYTE CORPORATION 发明人 RODGERS, JAMES, D
分类号 C07D487/04;A61K31/519 主分类号 C07D487/04
代理机构 代理人
主权项
地址