发明名称 Efficient synthetic method for sumadain A and its derivatives
摘要 PURPOSE: A novel synthetic method for sumadain A or derivative thereof is provided to quickly and efficiently prepare sumadain A and derivative thereof with excellent physiological activity. CONSTITUTION: A method for synthesizing sumadain A or derivative thereof comprises: a step of cyclizing 2,4,6-trihydroxyacetopenone and alpha,beta-unsaturated aldehyde under the presence of diacetate at 90-110°C for 8-12 hours; and a step of performing aldole condensation reaction of the reactant with benzaldehyde at room temperature for 42-56 hours. The sumadain A or derivative thereof is denoted by chemical formula 1 or 2.
申请公布号 KR101146826(B1) 申请公布日期 2012.05.21
申请号 KR20100000991 申请日期 2010.01.06
申请人 发明人
分类号 C07D493/04;C07D311/94 主分类号 C07D493/04
代理机构 代理人
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