发明名称 CRYSTALLINE 6,7-UNSATURATED-7-CARBAMOYL MORPHINANE DERIVATIVE, AND METHOD FOR PRODUCING SAME
摘要 The present invention provides a compound represented by Formula (IA): an acid addition salt thereof, and/or stable crystals of solvates thereof. The crystals are extremely useful as an active ingredient for producing pharmaceutical products. The present invention further provides a novel method for producing a 6,7-unsaturated-7-carbamoyl morphinane derivative.
申请公布号 WO2012063933(A1) 申请公布日期 2012.05.18
申请号 WO2011JP76034 申请日期 2011.11.11
申请人 SHIONOGI & CO., LTD.;TAMURA, YOSHINORI;NOGUCHI, KOUICHI;INAGAKI, MASANAO;MORIMOTO, KENJI;HAGA, NOBUHIRO;ODA, SHINICHI;OMURA, SOHEI 发明人 TAMURA, YOSHINORI;NOGUCHI, KOUICHI;INAGAKI, MASANAO;MORIMOTO, KENJI;HAGA, NOBUHIRO;ODA, SHINICHI;OMURA, SOHEI
分类号 C07D489/08;A61K31/485;A61P1/08;A61P1/10;B01J27/10;C07D271/06 主分类号 C07D489/08
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