发明名称 QUINAZOLINONE DERIVATIVES EFFECTIVE AS VANILLOID ANTAGONISTS
摘要 FIELD: medicine, pharmaceutics. ^ SUBSTANCE: invention refers to applying a quinazolinone compound of formula: wherein R3 has the values presented in the description and the patent claim, in the free form or in the form of salt. Also, the invention refers to a pharmaceutical composition exhibiting vanilloid receptor antagonist activity on the basis of said compounds. ^ EFFECT: there are produced new compounds and pharmaceutical composition on their basis which can find application in medicine for treating and preventing pain, gastrointestinal disorder. ^ 12 cl, 30 ex
申请公布号 RU2449995(C2) 申请公布日期 2012.05.10
申请号 RU20100112450 申请日期 2005.06.08
申请人 NOVARTIS AG 发明人 RITCHI TIMOTI DZHON;KALSHO EHNDR'JU DZHEJMS;BREJN KRISTOFER TOMAS;DZJADULEVICH EHDUARD KAROL;KHART TERENS
分类号 A61K31/505;A61K31/517;A61P29/00;C07D239/88;C07D239/91;C07D401/04 主分类号 A61K31/505
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