发明名称 NAPHTHYRIDIN-2 (1 H)-ONE COMPOUNDS USEFUL AS ANTIBACTERIALS
摘要 Compounds of Formula (I), wherein substituents R1, R2 and R5 are as defined, and Ar represents substituted phenyl, pyridyl, pyridazinyl, pyrimidinyl, pyrazinyl, thiazolyl, furanyl, imidazolyl and thiophenyl substituted by a hydroxyalkyl substituent and an optional other substituent; compositions containing them, their use in therapy, including their use as antibacterials, for example in the treatment of tuberculosis, and methods for the preparation of such compounds, are provided.
申请公布号 US2012115899(A1) 申请公布日期 2012.05.10
申请号 US201013144507 申请日期 2010.01.15
申请人 ALEMPARTE-GALLARDO CARLOS;BARROS-AGUIRRE DAVID;CACHO-IZQUIERDO MONICA;FIANDOR ROMAN JOSE MARIA;LAVANDERA DIAZ JOSE LUIS;REMUINAN-BLANCO MODESTO JESUS 发明人 ALEMPARTE-GALLARDO CARLOS;BARROS-AGUIRRE DAVID;CACHO-IZQUIERDO MONICA;FIANDOR ROMAN JOSE MARIA;LAVANDERA DIAZ JOSE LUIS;REMUINAN-BLANCO MODESTO JESUS
分类号 A61K31/4545;A61P31/04;A61P31/06;C07D471/04 主分类号 A61K31/4545
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