发明名称 NEW CLASS OF HISTONE DEACETYLASE INHIBITORS
摘要 This invention is related to new histone deacetylase inhibitors according to the general formula (I) wherein: Q is a bond, CH2, NR5 or oxygen, X is CH or nitrogen, Y is a bond, CH2, oxygen or NR6, Z is CH or nitrogen, R1, R2 are, independently, hydrogen or C1-C6 alkyl, R3, R4 are, independently, hydrogen, halogen, C1-C6 alkyl, C1-C6 alkoxy, C1-C6 haloalkyl or C1-C6 haloalkoxy, and R5 and R6 are as further defined in the specification, and pharmaceutical acceptable salts thereof.
申请公布号 US2012115867(A1) 申请公布日期 2012.05.10
申请号 US201113100670 申请日期 2011.05.04
申请人 MINUCCI SAVERIO;PELICCI PIER GIUSEPPE;MAI ANTONELLO;BALLARINI MARCO;GARGIULO GAETANO;MASSA SILVIO;THALER FLORIAN;PAIN GILLES;COLOMBO ANDREA;GAGLIARDI STEFANIA;VARASI MARIO;MERCURIO CIRO;DAC S.R.L. 发明人 MINUCCI SAVERIO;PELICCI PIER GIUSEPPE;MAI ANTONELLO;BALLARINI MARCO;GARGIULO GAETANO;MASSA SILVIO;THALER FLORIAN;PAIN GILLES;COLOMBO ANDREA;GAGLIARDI STEFANIA;VARASI MARIO;MERCURIO CIRO
分类号 A61K31/495;A61K31/496;A61K31/5377;A61P35/00;C07D295/155;C07D401/10;C07D413/06 主分类号 A61K31/495
代理机构 代理人
主权项
地址