发明名称 PROCESSES FOR THE PREPARATION OF 5-HT2C RECEPTOR AGONISTS
摘要 <p>The present invention relates to processes and intermediates useful in the preparation of (R)-8-chloro-l-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine (lorcaserin), a serotonin (5-?T) receptor modulator that is useful in the treatment of, for example, central nervous system disorders, such as obesity.</p>
申请公布号 WO2010148207(A3) 申请公布日期 2012.05.10
申请号 WO2010US39004 申请日期 2010.06.17
申请人 ARENA PHARMACEUTICALS, INC.;DEMATTEI, JOHN, A.;CARLOS, MARLON;CASTRO, RYAN, O.;CHUANG, TSUNG-HSUN;HADD, MARK, ALLEN;LU, XIAO-XIONG;MACIAS, MARK;SHAW, STEPHEN, M. 发明人 DEMATTEI, JOHN, A.;CARLOS, MARLON;CASTRO, RYAN, O.;CHUANG, TSUNG-HSUN;HADD, MARK, ALLEN;LU, XIAO-XIONG;MACIAS, MARK;SHAW, STEPHEN, M.
分类号 C07C17/16;C07C209/08;C07C209/74;C07C211/29 主分类号 C07C17/16
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