发明名称 |
Indazoles, benzisoxazoles and benzisothiazoles and their use as estrogenic agents |
摘要 |
The present invention relates to compounds of formula (I): in which R1, R2, R3, X, Y and A are as defined in the specification. The compounds are modulators of the estrogen receptors. |
申请公布号 |
US8173679(B2) |
申请公布日期 |
2012.05.08 |
申请号 |
US201113152433 |
申请日期 |
2011.06.03 |
申请人 |
RONDOT BENOIT;LAFAY JEAN;BONNET PAULE;CLERC THIERRY;DUC IGOR;DURANTI ERIC;PUCCIO FRANCOIS;SHIELDS JACQUELINE;BLOT CHRISTIAN;MAILLOS PHILIPPE;LABORATOIRE THERMAMEX |
发明人 |
RONDOT BENOIT;LAFAY JEAN;BONNET PAULE;CLERC THIERRY;DUC IGOR;DURANTI ERIC;PUCCIO FRANCOIS;SHIELDS JACQUELINE;BLOT CHRISTIAN;MAILLOS PHILIPPE |
分类号 |
A61K31/454;A61K31/416;A61K31/423;A61K31/428;C07D231/56;C07D261/20;C07D275/04;C07D401/06;C07D413/12 |
主分类号 |
A61K31/454 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|