发明名称 Quinazolinone derivatives as tubulin polymerization inhibitors
摘要 The present invention provides compounds of formula (I), their use as inhibitors of tubulin polymerization as well as pharmaceutical compositions comprising said compounds of formula (I) wherein R1, R2, R3, R4, R5, R6, n, m and X have defined meanings.
申请公布号 US8168644(B2) 申请公布日期 2012.05.01
申请号 US20090934733 申请日期 2009.03.26
申请人 FREYNE EDDY JEAN EDGARD;MEVELLEC LAURENCE ANNE;VIALARD JORGE EDUARDO;MEYER CHRISTOPHE;PASQUIER ELISABETH THERESE JEANNE;BOURDREZ XAVIER MARC;ANGIBAUD PATRICK RENE;JANSSEN PHARMACEUTICA NV 发明人 FREYNE EDDY JEAN EDGARD;MEVELLEC LAURENCE ANNE;VIALARD JORGE EDUARDO;MEYER CHRISTOPHE;PASQUIER ELISABETH THERESE JEANNE;BOURDREZ XAVIER MARC;ANGIBAUD PATRICK RENE
分类号 A01N43/54;A61K31/517;C07D239/72 主分类号 A01N43/54
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