发明名称 BICYCLOESTER DERIVATIVE
摘要 <p>SUMMARY Novel bicycloester derivatives and pharmaceutically acceptable salts thereof have high DPP-IV inhibitory activity. SOLVING MEANS The novel bicycloester derivatives are represented by the general formula (1): Pharmaceutically acceptable salts thereof are also included (Example: (2S,4S)-1-[[N-(4-ethoxycarbonylbicyclo[2.2.2]oct-1-yl)amino]acetyl]-4-fluoropyrrolidine-2-carbonitrile)).</p>
申请公布号 SI1712547(T1) 申请公布日期 2012.04.30
申请号 SI20050031480T 申请日期 2005.02.01
申请人 KYORIN PHARMACEUTICAL CO., LTD. 发明人 FUKUDA YASUMICHI;ASAHINA YOSHIKAZU;OHATA KOHEI;YOKOTA KAZUYA;MURAKAMI KOJI;MATSUI TOSHIYUKI
分类号 A61K31/40;A61K31/4025;A61P3/10;A61P43/00;C07D207/16;C07D405/12 主分类号 A61K31/40
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