发明名称 CO-CRYSTALS OF VX-950 (TELAPREVIR) OTHER COMPONENTS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME
摘要 Disclosed is a co-crystal comprising a compound of formula I (commonly known as telaprevir or VX-950) and a co-crystal former selected from the group consisting of 3-methoxy-4-hydroxybenzoic acid, 2,4-dihydroxybenzoic acid, and 2,5-dihydroxybenzoic acid.
申请公布号 NZ583699(A) 申请公布日期 2012.04.27
申请号 NZ20080583699 申请日期 2008.08.29
申请人 VERTEX PHARMACEUTICALS, INC. 发明人 ZHANG, YUEGANG;CONNELLY, PATRICK R;JOHNSTON, STEVE
分类号 C07D403/12;A61K31/454;A61P1/16 主分类号 C07D403/12
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