发明名称 |
CO-CRYSTALS OF VX-950 (TELAPREVIR) OTHER COMPONENTS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME |
摘要 |
Disclosed is a co-crystal comprising a compound of formula I (commonly known as telaprevir or VX-950) and a co-crystal former selected from the group consisting of 3-methoxy-4-hydroxybenzoic acid, 2,4-dihydroxybenzoic acid, and 2,5-dihydroxybenzoic acid.
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申请公布号 |
NZ583699(A) |
申请公布日期 |
2012.04.27 |
申请号 |
NZ20080583699 |
申请日期 |
2008.08.29 |
申请人 |
VERTEX PHARMACEUTICALS, INC. |
发明人 |
ZHANG, YUEGANG;CONNELLY, PATRICK R;JOHNSTON, STEVE |
分类号 |
C07D403/12;A61K31/454;A61P1/16 |
主分类号 |
C07D403/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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